阿拉丁小分子抑制劑、激動劑、拮抗劑--G蛋白偶聯受體信號通路(上)-自主發布-資訊-生物在線

阿拉丁小分子抑制劑、激動劑、拮抗劑--G蛋白偶聯受體信號通路(上)

作者:上海阿拉丁生化科技股份有限公司 2020-07-10T17:09 (訪問量:7755)

box-sizing: border-box;">M129297Mirtazapine≥98%85650-52-8100mg,1g5-HTSB742457SB742457≥97%607742-69-85mg,25mg5-HT69.63B129690BRL-15572≥99%193611-72-25mg,10mg,50mg 5-HT1D7.9P129785PRX-08066 Maleic acid≥99%866206-55-55mg,10mg,50mg 5-HT2B3.4 nMT124762鹽酸托烷司瓊≥98.0%105826-92-4250mg,1g,5g5-HT370.1±0.9 nMP129438Pizotifen Malate≥99%5189-11-7 100mg,500mg A129701Azasetron HCl≥99%123040-16-425mg,100mg5-HT30.33 nMF129636夫洛丙酮≥99%2295-58-150mg5-HT1AO129694Ondansetron≥99%99614-02-510mg,50mg,250mg 5-HT3P129744Palonosetron HCl≥99%135729-62-3100mg,500mg 5-HT3V129763VUF 10166≥99%155584-74-010mg,50mg,250mg5-HT3A0.04 nM5-HT3AB22 nMN159830奈法唑酮鹽酸鹽98.00%82752-99-6200mg,1gC101491鹽酸賽庚啶98%41354-29-41g,5g,25g5-HT20.6 nMO129679Ondansetron Hydrochloride Dihydrate≥98% (HPLC)103639-04-91g,5g5-HT3 receptor 6.16 nMA135530Alosetron Hydrochloride≥98% (HPLC)122852-69-11g,5g5-HT3 receptor S132232Sarpogrelate Hydrochloride≥98%135159-51-25mg,25mg,100mg5-HT2A8.525-HT2C7.435-HT2B6.57R166990Ramosetron hydrochloride98% (HPLC)132907-72-310mg,50mg,100mg,250mg 5-HT3 receptor 0.091 nMP111270葛根素98%3681-99-01g,5g,25g,100g 5-HT2CP111269葛根素分析標準品,≥98%3681-99-020mg5-HT2CC134704Cyclobenzaprine hydrochloride98%6202-23-91g,5g,25g5-HT2 receptor G127257Granisetron-109889-09-025mg,50mg,100mg,250mg 5HT-3L129692LY310762≥95%192927-92-710mg,50mg5-HT1D249 nMP125293Palonosetron-135729-61-210mg,100mg5-HT3 receptor 0.17 nMM1245745-甲氧基色胺97%608-07-1250mg,1g,5g,25g5-HT15-HT25-HT45-HT6S129681Sumatriptan Succinate≥98% (HPLC)103628-48-450mg,100mg,250mg,1g P129662Prucalopride≥99%179474-81-810mg,50mg5-HT4A2.5 nM5-HT4B8 nMA124880 Aripiprazole≥99%129722-12-91g,5g5-HT1A4.2 nMN129630 Naratriptan hydrochloride≥98%143388-64-110mg,25mg,50mg,100mg 5-HT R129638Rizatriptan Benzoate≥98%(HPLC)145202-66-010mg,50mg,250mg,1g,5g 5-HT1Z129649Zolmitriptan≥98%(HPLC)139264-17-8200mg,250mg,1g,5g,25g 5-HTM129673Mosapride Citrate≥98%112885-42-410mg,50mg,250mg,1g,5g,25g 5-HT4E129729Eletriptan HBr≥98%177834-92-310mg,50mg,250mg,1g,5g5-HT1B0.92 nM5-HT1D3.14 nMA129703Almotriptan Malate≥99%181183-52-81g5-HT1B5-HT1DT168187Tegaserod maleate98% (HPLC)189188-57-610mg,50mg5-HT4 receptor B129734BRL-54443≥98%57477-39-110mg,50mg,100mg5-HT1E8.75-HT1F9.25B178171 brexpiprazole97%913611-97-91gD2L0.3 nM5-HT1A0.12 nM5-HT2A0.47 nMα1B受體0.17 nMα2C受體0.59 nMM179481Mosapride95%112885-41-31g,5g5HT4S111161血清胺鹽酸鹽AR153-98-01g,5g,25g5-HTV124992Vilazodone≥98%163521-12-810mg,50mgF167802Flibanserin98% (HPLC)167933-07-55mg,25mg5-HT1A1 nM5-HT2A49 nMF167802Vortioxetine≥98%508233-74-710mg,50mg,250mg,1g P129402Azacyclonol≥99%115-46-850mg

*腎上腺素受體

項目號產品名稱規格CAS包裝靶點IC50KipKiKdEC50ED50pEC50
D129796甲磺酸多沙唑嗪≥99%77883-43-350mg,100mg,250mg,1g,5g,25g,100gα-1腎上腺素能受體
I129899Ivabradine HCl≥98%148849-67-6250mg,1g,5g腎上腺素受體2.9 μM
C129903Cisatracurium Besylate≥98%96946-42-81g腎上腺素受體
A124739Asenapine maleate≥98% (HPLC)85650-56-210mg,50mg,250mg,1g5-HT2C10.46
5-HT2A10.15
5-HT79.94
5-HT2B9.75
5-HT69.6
C141489卡拉洛爾98%57775-29-8250mg,1g
C120231 卡拉洛爾分析標準品57775-29-810mg
A129804Alfuzosin hydrochloride≥98%81403-68-150mg,100mg,250mg,1gα1受體
S126595Silodosin≥99%160970-54-75mg,25mg,100mg,250mg,1g
N129836Nebivolol hydrochloride≥97%152520-56-410mg,20mg,100mg,1g,5gβ1-腎上腺素受體0.8 nM
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